Elagolix Sodium 3.0

Elagolix Sodium 3.0Elagolix Soidum is a potent, selective, orally active, non peptide antagonist of the gonadotropin releasing hormone receptor (GnRHR) with Kd value of 54 pM. Concentration at 10 ? M shows no significant activity on ion channels, enzymes, and transporters (inhibition <50%).

the major stress hormone

ErbB2 and ErbB3 with IC50 of 4 nM

if the cylinder upsets

10-fold selective for B-RafV600E over wild-type B-Raf in enzymatic assays and the cellular selectivity can exceed 100-fold

Trichostatin A (TSA) is an HDAC inhibitor with IC50 of ~1

superoxide anion and ABTS radicals with anti-inflammatory

3081-200LO

Ranolazine is a calcium uptake inhibitor via the sodium/calcium channel

Corning These 22x450mm PYREX® Flash columns are ideal for use when quick separations in absorption chromatography applications are desired

Abacavir is a commonly used nucleoside analogue with potent antiviral activity against HIV-1

Probucol is an anti-hyperlipidemic drug by lowering the level of cholesterol in the bloodstream by increasing the rate of LDL catabolism

and does not inhibit closely related kinases MEK1